PHYSL 210A - ENDOCRINE

Created by Ameera Gani

Nervous system vs Endocrine system?
Endocrine is slower and more sustained control over long term processes

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TermDefinition
Nervous system vs Endocrine system?
Endocrine is slower and more sustained control over long term processes
What are the 2 glandular systems?
1. Exocrine glands: empty secretions into body cavities or onto body surfaces by tubular ducts 2. Endocrine glands: ductless glands that release secretions internally into bloodstream
What are the 2 types of hormones?
- Steroids: cholesterol - Proteins: amines, peptides
Do secretory vesicles expose hormones to proteolytic degradation?
No, they protect them from it
Secretory vesicles provide a _____ mechanism to the site of ______
- Transport (microtubules/microfilaments) - Release (plasma membrane)
What type of release mechanism do secretory vesicles use?
Exocytosis, vesicle is incorporated into plasma membrane
What are the 2 types of hormones in plasma?
- Bound - Free
Which hormone is biologically active?
Free
T/F: Plasma hormones are inactive when bound to binding protein
True
How does protein binding of plasma hormones provide a reservoir for target sites?
- Increase solubility/conc of lipid soluble and thyroid hormones
How does protein binding of plasma hormones protect hormones from degradation by liver/plasma enzymes?
By increasing size
How does protein binding of plasma hormones provide a buffer against changes in hormone conc?
By inactivating free hormones
Why is hormone secretion dynamically regulated?
Maintain steady state around range/point that varies w/ age
What happens when negative feedback of hormones takes place?
- Inhibits secretion when circulating levels are high - Increased secretion when circulating levels are low
What is the first requisite for hormonal action?
Binding of hormone to receptor
In the "Lock and Key" saying, what is the receptor and what is the hormone?
Lock: Receptor Key: Hormone
What are the 2 types of hormone receptors?
Nuclear and Cytoplasmic
What is the purpose of Nuclear receptors? 2
- Steroid/thyroid hormones - Genomically mediated through protein synthesis
What is the purpose of Cytoplasmic receptors? 2
- Intracellular T for cytosol-insoluble steroids - Reservoir storage and organelle actions for thyroid hormones
What happens during down regulation? 4
- At high hormone conc to prevent over-activity - Decreased receptor synthesis - Internalized membrane receptors - Dislocation of receptor system
What does desensitization/sensitization do to the Lock structure?
Conformational change in shape
What 2 things happen at high hormone conc to prevent over-activity?
- Down regulation (less receptors) - Desensitization (less affinity)
What happens during up regulation? 2
- At low hormone conc to increase activity - Increased receptor synthesis
What 2 things happen at to low hormone conc to increase activity?
- Up regulation (More receptors) - Sensitization (more affinity)
Why does down regulation happen with coated pits?
Allow proteins hormones to enter cell
What are 3 types of endocrine dysfunction?
1. Primary defect in synthesis 2. Defect in regulation 3. Defect in hormone action
Posterior pituary vs Anterior pituitary, which one has neural tissue?
Posterior P: neural tissue Anterior P: non-neural tissue (Rathke's pouch)
What are the posterior P hormones? 2
- ADH/vasopressin: SON - Oxytocin: PVN
What is the mechanism for vasoconstriction? 2
- Contract BV smooth muscle - Increase BP Only at high conc
What is the mechanism for ADH? 3
1. Increase permeability for renal collecting duct (increase # water channels) 2. VC reduces glomerular filtration rate 3. Contraction reduces size of glomerulosa cells = reduces SA for filtration
What are the 2 factors affecting secretion of ADH/vasopressin?
- Plasma volume - Plasma osmolarity
What is ADH secretion increased by? 4
- Stress - Heat - Nicotine - Caffeine
What is ADH secretion decreased by?
- Cold - Alcohol
What deficiency does problem with ADH production cause?
Hypothalamic/central diabetes insipidus
What deficiency does problem of ADH action cause?
Nephrogenic diabetes insipidus
How is syndrome of inappropriate ADH (SIADH) caused?
Problem of ADH production (feedback failure) - Excess
What is polyuria?
Large amounts of dilute urine
What is polydipsia?
Excessive thirst and fluid intake
How is the #/amp of growth hormone release episodes increased? 3
- Dark - Sleep - Fasting
T/F: Frequent meals high in glucose/FA increase growth hormone release?
False, it suppresses it
What is Type 1 dwarfism caused by?
Defect in GH production
What is laron-type dwarfism caused by? 3
- Defect in GH action - GH levels no deficient - IGF-1 levels are deficient
What are the components of sompatopause? 4
- GH deficiency in adults - Increased fat/decreased lean mass - Metabolic disturbance - Impaired immunity
What is acromegaly?
Excess GH production in adult
What are the actions of prolactin? 3
- Gonadal modulation: pro when gonadal acitivity is low - Mammary gland grows - Lactation
What are prolactin releasing factors? PRF 2
- TRH - Oxytocin
What are gonadal steroids for prolactin secretion? 2
- E/T increase - Progesterone decrease
What is Hyperprolactinemia? is there treatment?
Excess - Dopamine
What is Hypoprolactinemia?
Deficiency
What is hyperglycemia?
Pituitary diabetes - Excess
What is hypopituitarism?
Failure of P gland to produce hormones partially or completely
What is panhypopituitarism?
Absent production of all anterior pituitary hormones
What stimulates thyroid gland growth?
Peptide produced by pituitary thyrotrophs
What subunits are in the glycoprotein hormone?
Alpha & Beta
Where do biological activities happen in glycoprotein hormones?
In beta subunit
Where is thyroglobulin secreted and synthesized?
Synthesized: in rough ER of follicular cells Secreted: into colloid
What kind of residues does thyroglobulin provide a template for thyroid hormone synthesis?
Tyrosine
What is thyroxine (T4) converted to in peripheral tissues?
T3
Is T3 more or less biologically active than thyroxine?
More
T/F: thyroglobulin is a binding protein
False
What are the thyroid binding proteins? 3
- Thyroid-binding globulin - Thyroid binding albumin - Thyroid binding pre albumin
What is calorigenesis?
Increasing oxygen and glucose uptake by tissues - increase BMR
Is thyroid hormone action long or short responses?
Long
What is thyroid hormone effect on BMR?
Increase
What is thyroid hormone effect on heat production?
Increased O2 and glucose uptake = calorigenic effect = increased heat
What is thyroid hormones effect on neural activity?
Increased irritability and beta receptors, decreased reflex times
Does thyroid hormone increase or decrease plasma cholesterol?
Decrease
What 3 types of thyroid hormone receptors are there?
- Membrane bound - Cytoplasmic - Nuclear
What are membrane bound thyroid hormone receptors?
Linked to channels which allow glucose and O2 to be taken into cell
What are cytoplasmic thyroid hormone receptors?
Intracellular storage of TH or production of ATP in mito
What are nuclear thyroid hormone receptors?
Effect protein synthesis
T/F: TH's are hydrophobic
True, even though they contain tyrosine residues
What is caused by an excess in thyroid excess?
Hyperthyroidism
What is graves disease cause by?
LATS antibodies against the TSH receptor
What is caused by a deficiency in thyroid hormone?
Hypothyroidism
Does hypothyroidism cause an increase or decrease in BMR?
Decrease
What is an endemic goitre?
Iodine deficiency - decreased T3 and increased TSH
What does hashimoto's thyroiditis cause?
Antibodies against T3 or T4 or thyroglobulin
What is a thyroid hormone deficiency in utero called?
Cretinism - stunts metal and physical development
What is the buildup of hyaluronic acid and mucus edema under the skin called?
Myxedema
What is ACTH produced by?
Produced pituitary corticotrophs
What does ACTH stimulate?
Adrenal BF, growth and steroidogenesis
What zone is aldosterone in?
Glomerulosa
What does angiotensis II stimulate?
Alodesterone release from adrenal cortex in response to decreased ECF volume/low blood [Na]
What is intermediary metabolism?
Increased blood glucose through anabolic effects on liver and catabolic effects on other tissues
What does intermediary metabolism do for gluconeogenesis?
Stimulate it in the liver (anabolic)
What does intermediary metabolism do for triglyceride breakdown?
Stimulates it in adipose tissue w/ glycerol and FA release into blood (catabolic)
What does intermediary metabolism do for skin breakdown?
Stimulates it and breaks down connective tissue and muscle to release AA (catabolic)
Does glucocorticoid increased or decrease substrate availability?
Increase (increase tissue catabolism, decrease synthesis)
Does glucocorticoid increased or decrease substrate uptake by the liver?
Increase
Does glucocorticoid increased or decrease gluconeogensic enzymes?
Increase
Does glucocorticoid increased or decrease glycogenolysis?
Increased
What does cortisol do? 3
- Prevent inflammation - Prevent autoimmunity - Mobilize glucose
Where is DHEA (adrenal androgen) synthesized?
Zone reticularis
What are adrenal androgens converted to?
Testosterone and estrogen
What is adrenogenital syndrome?
Excess androgens from adrenal cortex
What are the 2 hypercalcemic hormones?
- Parathyroid hormone (PTH) - Vitamin D (VD)
What is the hypocalcemic hormone?
Calcitonin (CT)
What does PTH do to plasma Calcium and Phosphate?
- Ca: Increase - PO4: Decrease
What does PTH do to Ca, PO4, and VD in the kidney?
- Ca: increase reabsorption - PO4: decrease reabsorption - VD: increase activation
What does PTH do to bones?
Increase bone resorption
What effect does PTH have on GIT?
Increase VD formation
What inhibits PTH secretion? Hypercalcemia or Hypocalcemia?
Hypercalcemia inhibits Hypocalcemia stimulates
Where does PTH come from?
Parathyroid gland (chief cells)
What 3 things does Hyperparathyroidism affect?
Bones Stones Abdominal groans
What does Hyperparathyrodism do to PTH, Ca, PO4, and VD?
- PTH, Ca, VD: increase - PO4: decrease
What is the "stones" part of hyperparathyroidism?
Soft tissue calcification = Kidney stones
What is the "bones" part of hyperparathyroidism?
Weak bones, fractures (bone resorption)
What is the "abdominal groans" part of hyperparathyroidism?
GIT dysfunction
What are the Ca levels of kidney stones?
10-12 mg/dL
What is Ca levels of death?
17 mg/dL
What are the effects on Ca and PO4 during secondary hyperparathyroidism?
Ca: Decrease PO4: increase
What are the effects on Ca and VD during secondary hyperparathyroidism in rickets?
Impaired GI uptake of Ca Decreased VD
What are the effects on Ca during secondary hyperparathyroidism in renal failure?
Impaired renal reabsorption of Ca
What are the effects on PTH, Ca, PO4, and VD during primary hypoparathyroidism?
PTH, Ca, VD: Decrease PO4: increase
What is primary hypoparathyroidism's effect on neuromuscular activity?
Decreased Ca = decreased threshold for excitation = repetitive responses
What is trousseau's sign?
Involuntary contraction of carpal muscle due to hypocalcemia and tetany - Hypoparathyroidism
What are the effects on PTH, Ca, PO4, and VD during pseudohypoparathyroidism?
PTH, PO4, VD: increase Ca: decrease
What are C-cells?
Parafollicular cells - Release calcitonin - Peptide hormone
What are the effects of calcitonin on plasma Ca and PO4?
Decrease both
What are the effects of calcitonin on Ca, PO4, and VD in the kidney?
Decrease all reabsorption/activation
What are the effects of calcitonin on bones?
Decreased bone resorption
What is the stimulus for calcitonin secretion?
Increased plasma Ca
What are the effects of VD on plasma Ca and PO4?
Increase both
What are the effects of VD on Ca and PO4 in the kidney?
Increase both reabsorption
What is the effect of VD on bones?
Promote PTH actions
What does a deficiency in VD cause?
- Rickets in juvenils - Osteomalacia in adults
What is sympathetic stimulation for glucagon and insulin?
Glucagon: Increase Insulin: Decrease
What is parasympathetic stimulation for glucagon and insulin?
Glucagon: Increase Insulin: Increase
What is the purpose of insulin? Anabolic or catabolic?
- Convert nutrients into stored forms to lower blood glucose - Anabolic
What is the purpose of glucagon? anabolic or catabolic?
- Breakdown stored forms of energy to increase blood glucose - Catabolic
What are glucagon effects on glucose for glycogenesis, gluconeogenesis, glycogenolysis?
Glycogenesis: decrease Gluconeogenesis & glycogenolysis: increase
What are glucagon effects on lipids for lipolysis and lipogenesis?
Lipolysis: increase Lipogenesis: decrease
Is diabetes mellitus a glucagon deficiency or excess?
Excess; insulin deficiency
What is type I diabetes?
- Beta cells destructed = decreased insulin release
What is type II diabetes?
- target cells have decreased response to insulin